SCHEMBL7861824

SCHEMBL7861824

CC(C)(C)OC(=O)Nc1cccc(OCCN)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.50
PLAU P00749 2/20 0.49
THRB P10828 1/20 0.48
BRAF P15056 1/20 0.47
EGFR P00533 2/20 0.46
ITK Q08881 2/20 0.46
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
SYK P43405 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
AURKA O14965 1/20 0.44
RPS6KB1 P23443 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24861173 0.93 FAAH (0.46) FAAHPLAUTHRBBRAFEGFR
SCHEMBL29024421 0.93 FAAH (0.46) FAAHPLAUTHRBBRAFEGFR
SCHEMBL595191 0.88 FAAH (0.51) FAAHTHRBEGFRITKMAPT
SCHEMBL6470099 0.87 FAAH (0.66) FAAHTHRBMAPTSMN1; SMN2MEN1
SCHEMBL21768037 0.87 THRB (0.51) FAAHTHRBMAPTSMN1; SMN2MEN1
SCHEMBL6470532 0.85 HTT (0.58) FAAHPLAUTHRBMAPTSMN1; SMN2
SCHEMBL6595861 0.84 FAAH (0.50) FAAHTHRBEGFRITKMAPT
SCHEMBL12519749 0.84 FAAH (0.50) FAAHTHRBEGFRITKMAPT
SCHEMBL7103629 0.83 ALDH1A1 (0.50) FAAHMAPTSYKMEN1KMT2A
SCHEMBL480266 0.83 MAPK1 (0.61) MAPTSMN1; SMN2MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067928-A4 METHODS FOR INHIBITING MRP1 LILLY CO ELI (US) 2001-11-14 EP disclosed
EP-1067928-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 2001-01-17 EP disclosed
WO-1999051228-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 1999-10-14 WO disclosed