SCHEMBL7103629

SCHEMBL7103629

CC(C)(C)OC(=O)Nc1cccc(OC(=O)CCN)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
CYP3A4 P08684 2/20 0.50
FAAH O00519 1/20 0.50
MAPK1 P28482 1/20 0.50
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
MAPT P10636 3/20 0.44
TDP2 O95551 1/20 0.43
HDAC3 O15379 4/20 0.43
HDAC1 Q13547 3/20 0.43
HDAC2 Q92769 3/20 0.43
GAA P10253 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GLA P06280 1/20 0.43
HPGD P15428 1/20 0.43
HIF1A Q16665 1/20 0.43
CYP17A1 P05093 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25736700 0.89 ALDH1A1 (0.49) ALDH1A1CYP3A4FAAHMAPK1CA1
SCHEMBL25736723 0.86 CYP3A4 (0.51) ALDH1A1CYP3A4FAAHMAPK1RXFP1
SCHEMBL7861824 0.83 FAAH (0.50) FAAHMAPTHDAC3HDAC1HDAC2
SCHEMBL999347 0.82 KMT2A (0.61) ALDH1A1CYP3A4FAAHMAPK1RXFP1
SCHEMBL3892771 0.82 ALDH1A1 (0.52) ALDH1A1CYP3A4FAAHMAPK1CA1
SCHEMBL2348855 0.81 ALDH1A1 (0.42) ALDH1A1CYP3A4FAAHMAPK1CA1
SCHEMBL2348861 0.81 ALDH1A1 (0.42) ALDH1A1CYP3A4FAAHMAPK1CA1
SCHEMBL2222285 0.81 ALDH1A1 (0.42) ALDH1A1CYP3A4FAAHMAPK1CA1
SCHEMBL26785208 0.80 MAPK1 (0.50) ALDH1A1CYP3A4FAAHMAPK1CA1
SCHEMBL27373863 0.80 MTNR1B (0.45) ALDH1A1CYP3A4FAAHMAPK1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030162799-A1 Carbocyclic oxo, carboxy amines such as 3-(4-(3,5-Dichloro-4-pyridylcarboxamido)phenyl)-2-(2-propylamino-3,4 -dioxocyclobut-1-enyl)amino)propanoic acid, used as integrin antagonists; antiinflammatory agents CELLTECH R&D LIMITED (GB) 2003-08-28 US disclosed
US-6518283-B1 To modify integrin function in such a way as to beneficially modulate cell adhesion CELLTECH R&D LIMITED (GB) 2003-02-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030162799-A1 Carbocyclic oxo, carboxy amines such as 3-(4-(3,5-Dichloro-4-pyridylcarboxamido)phenyl)-2-(2-propylamino-3,4 -dioxocyclobut-1-enyl)amino)propanoic acid, used as integrin antagonists; antiinflammatory agents ICAM1, VCAM1, CCR1 ALDH1A1 287/4885CYP3A4 4086/4885FAAH 1097/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.