SCHEMBL7861992

SCHEMBL7861992

CC(=O)N[C@@H](Cc1cccc(CNC(=O)c2cccc(NC(=N)N)c2)c1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.52
ITGAV P06756 3/20 0.52
ITGA2B P08514 2/20 0.52
ITGB1 P05556 1/20 0.52
ITGB5 P18084 1/20 0.52
GRB2 P62993 1/20 0.48
ALDH1A1 P00352 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CHRM3 P20309 1/20 0.46
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
BCHE P06276 1/20 0.45
SENP1 Q9P0U3 3/20 0.45
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
PLAU P00749 1/20 0.43
PLAUR Q03405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864217 1.00 ITGB3 (0.52) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7862001 0.85 ITGB3 (0.48) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7861998 0.85 ITGB3 (0.48) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7377320 0.85 ITGB1 (0.70) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7377326 0.85 ITGB1 (0.70) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8499774 0.85 SENP1 (0.42) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL20999541 0.80 ITGB1 (0.54) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7856474 0.80 SIRT2 (0.51) ALDH1A1L3MBTL1LMNAMAPK1BCHE
SCHEMBL7374891 0.79 ITGB1 (0.57) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7378081 0.79 ITGB1 (0.57) ITGB3ITGAVITGA2BITGB1ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP disclosed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed