SCHEMBL7864170

SCHEMBL7864170

CCOC(=O)C(Cc1cccc(CNC(=O)c2cccc(NC=NN)c2)c1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.47
PPARG P37231 3/20 0.47
LMNA P02545 2/20 0.42
MAPK1 P28482 1/20 0.42
ALDH1A1 P00352 3/20 0.41
HTT P42858 2/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.41
BCHE P06276 2/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PKM P14618 1/20 0.40
CFD P00746 1/20 0.40
SENP1 Q9P0U3 2/20 0.40
SENP2 Q9HC62 1/20 0.40
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864788 0.90 SIRT2 (0.44) EPHX2PPARGLMNAMAPK1ALDH1A1
SCHEMBL7863145 0.87 EPHX2 (0.54) EPHX2PPARGLMNABCHE
SCHEMBL7862057 0.86 ALDH1A1 (0.41) EPHX2PPARGLMNAALDH1A1PKM
SCHEMBL7861967 0.84 NAMPT (0.54) EPHX2PPARGLMNAMAPK1ALDH1A1
SCHEMBL7864776 0.82 PPARG (0.53) EPHX2PPARGLMNABCHE
SCHEMBL7864267 0.82 TP53 (0.45) PPARGLMNAMAPK1ALDH1A1HTT
SCHEMBL7862050 0.81 PPARG (0.44) EPHX2PPARGLMNAMAPK1ALDH1A1
SCHEMBL7856483 0.80 SIRT2 (0.48) EPHX2PPARGLMNAMAPK1ALDH1A1
SCHEMBL7864712 0.80 SIRT2 (0.45) EPHX2PPARGLMNAMAPK1ALDH1A1
SCHEMBL7825718 0.80 TP53 (0.47) ALDH1A1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed