SCHEMBL7862057

SCHEMBL7862057

CCOC(=O)C(Cc1cccc(CCc2cccc(NC=NN)c2)c1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
DHODH Q02127 2/20 0.41
CHRM1 P11229 1/20 0.41
EPHX2 P34913 1/20 0.39
PPARG P37231 1/20 0.39
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
F10 P00742 1/20 0.38
CTSB P07858 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MMP8 P22894 1/20 0.37
FFAR1 O14842 1/20 0.37
EPHX1 P07099 1/20 0.37
EGFR P00533 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7866946 0.88 EPHX1 (0.41) CTSBFFAR1EPHX1
SCHEMBL7864170 0.86 EPHX2 (0.47) ALDH1A1EPHX2PPARGLMNAPKM
SCHEMBL7864160 0.77 FFAR1 (0.39) LMNAFFAR1
SCHEMBL15553196 0.74 CHRM1 (0.66) ALDH1A1CHRM1EPHX2PPARGKDM4E
SCHEMBL7864788 0.74 SIRT2 (0.44) ALDH1A1EPHX2PPARGLMNA
SCHEMBL7452094 0.73 ITGB3 (0.48) ALDH1A1TP53LMNAPKMCA12
SCHEMBL30902537 0.73 NOS3 (0.60) PKMKDM4EEGFR
SCHEMBL7856489 0.72 ITGB3 (0.55) PPARGMMP8FFAR1MAPT
SCHEMBL7863145 0.72 EPHX2 (0.54) EPHX2PPARGLMNA
SCHEMBL7825718 0.72 TP53 (0.47) ALDH1A1TP53CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed