SCHEMBL7864280

SCHEMBL7864280

N=C(N)Nc1cccc(CC(=O)Nc2cccc(CCC(=O)O)c2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.62
ITGA2B P08514 1/20 0.62
ITGB1 P05556 1/20 0.55
ITGA4 P13612 1/20 0.55
SELP P16109 2/20 0.54
SELE P16581 2/20 0.54
SELL P14151 1/20 0.54
MAPT P10636 2/20 0.52
GAA P10253 1/20 0.52
GFER P55789 1/20 0.52
SIRT1 Q96EB6 1/20 0.51
CFD P00746 1/20 0.48
KMT2A Q03164 3/20 0.48
EPHX2 P34913 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.47
FFAR1 O14842 1/20 0.47
HTR1A P08908 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856482 0.87 ITGB3 (0.65) ITGB3ITGA2BITGB1ITGA4SELP
SCHEMBL23518466 0.85 ITGB3 (0.50) ITGB3ITGA2BSELPSELESELL
SCHEMBL7864626 0.84 SELP (0.54) ITGB3ITGA2BITGB1ITGA4SELP
SCHEMBL288541 0.84 ITGB3 (0.61) ITGB3ITGA2BSELPSELESELL
SCHEMBL7861970 0.84 ITGB3 (0.76) ITGB3ITGA2BITGB1SIRT1KMT2A
SCHEMBL8410309 0.83 ITGB3 (0.71) ITGB3ITGA2BITGB1ITGA4SELP
SCHEMBL7346500 0.83 ITGB3 (0.60) ITGB3ITGA2BITGB1MAPTGAA
SCHEMBL4407485 0.81 ATM (0.56) ITGB3ITGA2BSELPSELESELL
SCHEMBL7373162 0.81 HDAC3 (0.58) ITGB3ITGA2BITGB1ITGA4MAPT
SCHEMBL8371139 0.80 ITGB3 (0.57) ITGB3ITGA2BSIRT1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP disclosed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed