SCHEMBL7864636

SCHEMBL7864636

CCC(CC(=O)O)c1cccc(NS(=O)(=O)c2cccc(NC=NN)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.41
ITGB3 P05106 2/20 0.41
ITGAV P06756 2/20 0.41
PFKFB3 Q16875 1/20 0.40
F2 P00734 1/20 0.40
F10 P00742 1/20 0.40
PRSS1 P07477 1/20 0.40
CA1 P00915 4/20 0.39
CA2 P00918 4/20 0.39
CASP3 P42574 1/20 0.39
HTR6 P50406 3/20 0.38
POLB P06746 1/20 0.38
PTGES O14684 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7863259 0.86 PKM (0.46) PKMITGB3ITGAVF2F10
SCHEMBL7856452 0.83 PKM (0.43) PKMITGB3ITGAVF2F10
SCHEMBL7856455 0.83 PKM (0.43) PKMITGB3ITGAVF2F10
SCHEMBL8371142 0.83 PFKFB3 (0.43) PKMPFKFB3CA1CA2HTR6
SCHEMBL7864234 0.82 PGR (0.41) ITGB3ITGAVPFKFB3HTR6POLB
SCHEMBL7866912 0.82 SMN1; SMN2 (0.41) ITGB3ITGAVPFKFB3HDAC2HDAC8
SCHEMBL7861775 0.82 EEF2K (0.43) ITGB3ITGAVPFKFB3CA1CA2
SCHEMBL7864756 0.81 CA1 (0.38) PKMITGB3ITGAVPFKFB3CA1
SCHEMBL7864664 0.81 GBA1 (0.39) PKMITGB3ITGAVPFKFB3CA1
SCHEMBL7864164 0.80 HDAC4 (0.38) PKMITGB3ITGAVPFKFB3CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed