SCHEMBL7864756

SCHEMBL7864756

NN=CNc1cccc(S(=O)(=O)Nc2cccc(C(CC(=O)O)c3cc(F)c(F)c(F)c3)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
PFKFB3 Q16875 1/20 0.38
MAPT P10636 2/20 0.38
GBA1 P04062 1/20 0.38
HTR6 P50406 2/20 0.37
HSD17B1 P14061 4/20 0.37
HSD17B2 P37059 4/20 0.37
ITGB3 P05106 1/20 0.37
ITGAV P06756 1/20 0.37
LMNA P02545 2/20 0.37
TP53 P04637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GAA P10253 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
MPI P34949 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864664 0.91 GBA1 (0.39) CA1CA2PFKFB3MAPTGBA1
SCHEMBL7861775 0.91 EEF2K (0.43) CA1CA2PFKFB3MAPTGBA1
SCHEMBL7866912 0.89 SMN1; SMN2 (0.41) PFKFB3MAPTGBA1ITGB3ITGAV
SCHEMBL7864164 0.89 HDAC4 (0.38) CA1CA2PFKFB3MAPTGBA1
SCHEMBL7864234 0.87 PGR (0.41) PFKFB3HTR6ITGB3ITGAVMEN1
SCHEMBL7864212 0.86 MEN1 (0.41) CA1CA2MAPTGBA1HTR6
SCHEMBL7864636 0.81 PKM (0.41) CA1CA2PFKFB3HTR6ITGB3
SCHEMBL7864668 0.80 GAA (0.40) CA1CA2PFKFB3MAPTHTR6
SCHEMBL7863160 0.80 EEF2K (0.41) PFKFB3MAPTGBA1HTR6ITGB3
SCHEMBL7863156 0.80 EEF2K (0.41) PFKFB3MAPTGBA1HTR6ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed