SCHEMBL7864664

SCHEMBL7864664

NN=CNc1cccc(S(=O)(=O)Nc2cccc(C(CC(=O)O)c3c(F)c(F)cc(F)c3F)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.39
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
PFKFB3 Q16875 1/20 0.38
MAPT P10636 2/20 0.37
CA9 Q16790 1/20 0.37
HSD17B1 P14061 4/20 0.37
HSD17B2 P37059 4/20 0.37
CASP3 P42574 1/20 0.37
HTR6 P50406 2/20 0.36
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
LMNA P02545 2/20 0.36
TP53 P04637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GAA P10253 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864756 0.91 CA1 (0.38) GBA1CA1CA2PFKFB3MAPT
SCHEMBL7864164 0.88 HDAC4 (0.38) GBA1CA1CA2PFKFB3MAPT
SCHEMBL7856460 0.87 CA1 (0.41) GBA1CA1CA2MAPTCA9
SCHEMBL7866912 0.87 SMN1; SMN2 (0.41) GBA1PFKFB3MAPTITGB3ITGAV
SCHEMBL7861775 0.87 EEF2K (0.43) GBA1CA1CA2PFKFB3MAPT
SCHEMBL7864234 0.83 PGR (0.41) PFKFB3HTR6ITGB3ITGAVMEN1
SCHEMBL7864636 0.81 PKM (0.41) CA1CA2PFKFB3CASP3HTR6
SCHEMBL8371142 0.80 PFKFB3 (0.43) CA1CA2PFKFB3MAPTHTR6
SCHEMBL7864212 0.78 MEN1 (0.41) GBA1CA1CA2MAPTCA9
SCHEMBL7864668 0.78 GAA (0.40) CA1CA2PFKFB3MAPTHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed