SCHEMBL7864673

SCHEMBL7864673

CCC(CC(=O)O)c1cccc(CNC(=O)c2cc(NC=NN)cc(C(F)(F)F)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PLA2G1B P04054 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
TACR1 P25103 3/20 0.41
LMNA P02545 2/20 0.40
RAB9A P51151 1/20 0.40
MLYCD O95822 2/20 0.40
MAPK14 Q16539 1/20 0.39
BCHE P06276 1/20 0.38
NNMT P40261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864751 0.87 SIRT2 (0.41) HTTGAALMNAPPARG
SCHEMBL7864633 0.86 MAPT (0.41) MAPTMEN1KMT2AHTTNPSR1
SCHEMBL7856467 0.85 MEN1 (0.42) MAPTMEN1KMT2AHTTNPSR1
SCHEMBL7866898 0.78 ALDH1A1 (0.42) MAPTMEN1KMT2AHTTCYP1A2
SCHEMBL7856468 0.76 TP53 (0.46) MEN1KMT2AHTTGAALMNA
SCHEMBL7864712 0.74 SIRT2 (0.45) HTTGAALMNAEPHX2PPARG
SCHEMBL7864178 0.74 TP53 (0.43) GAALMNAPPARGCHRM3
SCHEMBL7862019 0.73 LMNA (0.45) MAPTHTTLMNABCHEPPARG
SCHEMBL7864322 0.73 AURKA (0.41) MAPTGAALMNAEPHX2PPARG
SCHEMBL7824080 0.71 ITGB3 (0.54) HTTTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed