SCHEMBL7866947

SCHEMBL7866947

NN=CNc1cccc(C#Cc2cccc(C(CC(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.41
FFAR1 O14842 3/20 0.39
CTSA P10619 3/20 0.37
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
MMP12 P39900 2/20 0.36
MMP14 P50281 1/20 0.36
MMP15 P51511 1/20 0.36
MMP16 P51512 1/20 0.36
MMP26 Q9NRE1 1/20 0.36
LMNA P02545 1/20 0.35
EEF2K O00418 1/20 0.35
ALOX5 P09917 1/20 0.35
EPHX2 P34913 1/20 0.35
CYP2C19 P33261 1/20 0.35
HPGDS O60760 1/20 0.34
MEN1 O00255 1/20 0.34
THRB P10828 1/20 0.34
KMT2A Q03164 1/20 0.34
HDAC8 Q9BY41 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864160 0.82 FFAR1 (0.39) FFAR1CTSALMNACYP2C19KMT2A
SCHEMBL7864754 0.82 PTPN11 (0.48) PTPN11FFAR1MMP2MMP9MMP12
SCHEMBL7866927 0.80 FFAR1 (0.45) FFAR1HDAC8
SCHEMBL7856436 0.80 ITGB3 (0.48) MEN1KMT2A
SCHEMBL7863159 0.79 KMT2A (0.56) FFAR1CTSAKMT2A
SCHEMBL7457204 0.77 ITGB3 (0.53) FFAR1LMNAMEN1KMT2AHDAC8
SCHEMBL7863123 0.77 ITGB3 (0.39) CTSALMNAMEN1KMT2A
SCHEMBL8501227 0.77 ITGB3 (0.40) FFAR1CTSA
SCHEMBL7864766 0.77 ITGB3 (0.38) FFAR1CTSACYP2C19MEN1KMT2A
SCHEMBL7864712 0.76 SIRT2 (0.45) LMNAEPHX2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed