SCHEMBL7864754

SCHEMBL7864754

N=C(N)Nc1cccc(C#Cc2cccc(C(CC(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.48
FFAR1 O14842 1/20 0.39
IKBKB O14920 3/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
LMNA P02545 1/20 0.38
ITGB3 P05106 4/20 0.38
ITGA2B P08514 4/20 0.38
KDR P35968 1/20 0.38
PARP1 P09874 1/20 0.37
PARP10 Q53GL7 1/20 0.37
ITGAV P06756 1/20 0.37
CASR P41180 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP12 P39900 1/20 0.36
MMP14 P50281 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7866947 0.82 PTPN11 (0.41) PTPN11FFAR1LMNACASRMMP2
SCHEMBL7863285 0.82 ITGB3 (0.48) POLBMAPTMAPK1LMNAITGB3
SCHEMBL7861944 0.81 HDAC1 (0.45) POLBMAPTMAPK1LMNAITGB3
SCHEMBL7856431 0.81 HDAC1 (0.45) POLBMAPTMAPK1LMNAITGB3
SCHEMBL7856433 0.81 ITGB3 (0.54) POLBMAPTITGB3ITGA2BPARP1
SCHEMBL7856428 0.80 PARP1 (0.44) POLBMAPTMAPK1LMNAITGB3
SCHEMBL7863273 0.79 FFAR1 (0.43) FFAR1POLBMAPTMAPK1LMNA
SCHEMBL7863151 0.79 KMT2A (0.57) FFAR1
SCHEMBL7455765 0.78 ITGB3 (0.58) POLBITGB3ITGA2BALDH1A1
SCHEMBL7862046 0.77 ITGB3 (0.45) POLBMAPTITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP disclosed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed