Benzenesulfonamide

Benzenesulfonamide

SCHEMBL7866959

NS(=O)(=O)c1ccccc1.O=S(=O)(Nc1c(-c2ccccc2)noc1CO)c1ccccc1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.63
CA1 P00915 6/20 0.48
CA2 P00918 6/20 0.48
CA9 Q16790 5/20 0.48
CA12 O43570 4/20 0.48
MT-CO2 P00403 3/20 0.48
CA4 P22748 2/20 0.48
CA7 P43166 2/20 0.48
LMNA P02545 1/20 0.48
CA3 P07451 1/20 0.48
ADRB2 P07550 1/20 0.48
ADRB1 P08588 1/20 0.48
CYP3A4 P08684 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
CHRM1 P11229 1/20 0.48
ADRA2B P18089 1/20 0.48
PTGS1 P23219 1/20 0.48
CA6 P23280 1/20 0.48
SLC6A2 P23975 1/20 0.48
PDE4A P27815 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8348668 0.94 PTGS2 (0.53) PTGS2MT-CO2PTGS1ALDH1A1NPSR1
SCHEMBL8477416 0.84 ALDH1A1 (0.47) PTGS2MT-CO2ALDH1A1NPSR1PKM
SCHEMBL8597059 0.84 PTGS2 (0.45) PTGS2MT-CO2ALDH1A1NPSR1PKM
SCHEMBL8476337 0.84 ALDH1A1 (0.49) PTGS2MT-CO2PTGS1ALDH1A1NPSR1
Benzenesulfonamide SCHEMBL7180310 0.83 PTGS2 (0.62) PTGS2CA1CA2CA9CA12
SCHEMBL8475895 0.82 PTGS2 (0.54) PTGS2MT-CO2PTGS1ALDH1A1NPSR1
SCHEMBL8473431 0.81 ALDH1A1 (0.51) PTGS2MT-CO2PTGS1ALDH1A1NPSR1
SCHEMBL8473498 0.81 ALDH1A1 (0.48) PTGS2MT-CO2PTGS1ALDH1A1NPSR1
SCHEMBL8474218 0.80 ALDH1A1 (0.50) PTGS2MT-CO2PTGS1ALDH1A1NPSR1
SCHEMBL8473748 0.79 ALDH1A1 (0.45) PTGS2MT-CO2ALDH1A1NPSR1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001527542-A 2001-12-25 JP claimed
EP-1140181-A1 COMBINATION THERAPY OF RADIATION AND A COX-2 INHIBITOR FOR THE TREATMENT OF NEOPLASIA G.D. SEARLE & CO. (US) 2001-10-10 EP claimed
WO-2000038716-A1 COMBINATION THERAPY OF RADIATION AND A COX-2 INHIBITOR FOR THE TREATMENT OF NEOPLASIA G.D. SEARLE & CO. (US) 2000-07-06 WO claimed
EP-0979077-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. Searle & Co. (US) 2000-02-16 EP claimed
WO-1998047509-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1998-10-29 WO claimed