SCHEMBL8348668

SCHEMBL8348668

O=S(=O)(Nc1c(-c2ccccc2)noc1CO)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.53
ALDH1A1 P00352 3/20 0.51
NPSR1 Q6W5P4 1/20 0.51
MT-CO2 P00403 2/20 0.48
PKM P14618 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
EDNRB P24530 5/20 0.45
EDNRA P25101 5/20 0.45
NR4A2 P43354 1/20 0.45
NR1I2 O75469 1/20 0.43
PTGS1 P23219 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzenesulfonamide SCHEMBL7866959 0.94 PTGS2 (0.63) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8597059 0.90 PTGS2 (0.45) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8476337 0.90 ALDH1A1 (0.49) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8475895 0.88 PTGS2 (0.54) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8477416 0.87 ALDH1A1 (0.47) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8473431 0.86 ALDH1A1 (0.51) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8474218 0.85 ALDH1A1 (0.50) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8473748 0.84 ALDH1A1 (0.45) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8478927 0.84 ALDH1A1 (0.49) PTGS2ALDH1A1NPSR1MT-CO2PKM
SCHEMBL8479939 0.84 ALDH1A1 (0.49) PTGS2ALDH1A1NPSR1MT-CO2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0941080-A2 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS AS ANTI-ANGIOGENIC AGENTS G.D. SEARLE & CO. (US) 1999-09-15 EP disclosed
US-5932598-A NOVEL SUBSTITUTED SULFONAMIDE COMPOUNDS USEFUL AS PRODRUGS; ADMINISTERING TO TREAT INFLAMMATION-ASSOCIATED PAIN DUE TO CANCER, DENTAL PAIN; CYCLOOXYGENASE-2 INHIBITORS G. D. SEARLE & CO. (US) 1999-08-03 US disclosed
US-5859257-A ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS G. D. SEARLE & CO. (US) 1999-01-12 US disclosed
WO-1998022101-A2 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS AS ANTI-ANGIOGENIC AGENTS G.D. SEARLE & CO. (US) 1998-05-28 WO disclosed