SCHEMBL8476337

SCHEMBL8476337

O=S(=O)(Nc1c(-c2ccccc2)noc1CCO)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
NPSR1 Q6W5P4 1/20 0.49
PTGS2 P35354 6/20 0.46
MT-CO2 P00403 2/20 0.46
PKM P14618 1/20 0.44
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
NR4A2 P43354 1/20 0.43
EDNRB P24530 5/20 0.43
EDNRA P25101 5/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
NR1I2 O75469 1/20 0.41
PTGS1 P23219 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8477416 0.93 ALDH1A1 (0.47) ALDH1A1NPSR1PTGS2MT-CO2PKM
SCHEMBL8348668 0.90 PTGS2 (0.53) ALDH1A1NPSR1PTGS2MT-CO2PKM
SCHEMBL8474218 0.88 ALDH1A1 (0.50) ALDH1A1NPSR1PTGS2MT-CO2PKM
SCHEMBL8473498 0.86 ALDH1A1 (0.48) ALDH1A1NPSR1PTGS2MT-CO2PKM
SCHEMBL8475895 0.85 PTGS2 (0.54) ALDH1A1NPSR1PTGS2MT-CO2PKM
SCHEMBL8473748 0.84 ALDH1A1 (0.45) ALDH1A1NPSR1PTGS2MT-CO2PKM
SCHEMBL8473431 0.84 ALDH1A1 (0.51) ALDH1A1NPSR1PTGS2MT-CO2PKM
Benzenesulfonamide SCHEMBL7866959 0.84 PTGS2 (0.63) ALDH1A1NPSR1PTGS2MT-CO2PKM
SCHEMBL8476782 0.83 ALDH1A1 (0.46) ALDH1A1NPSR1PTGS2MT-CO2PKM
SCHEMBL8478927 0.82 ALDH1A1 (0.49) ALDH1A1NPSR1PTGS2MT-CO2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5700816-A ANTIARTHRITIC AGENTS G.D. SEARLE & CO. 1997-12-23 US claimed
US-5859257-A ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS G. D. SEARLE & CO. (US) 1999-01-12 US disclosed
US-5700816-A ANTIARTHRITIC AGENTS G.D. SEARLE & CO. 1997-12-23 US disclosed