SCHEMBL7867597

SCHEMBL7867597

Cc1cc(-c2ccccc2COc2ccccc2)ccc1[C@@H]1CCCNC1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.46
CHRNA4 P43681 1/20 0.46
SLC6A2 P23975 2/20 0.46
SLC6A4 P31645 2/20 0.46
SLC6A3 Q01959 2/20 0.46
PRMT5 O14744 2/20 0.44
FFAR4 Q5NUL3 2/20 0.42
PTGER1 P34995 1/20 0.42
PTGER4 P35408 1/20 0.42
PTGER3 P43115 1/20 0.42
PTGER2 P43116 1/20 0.42
HTR6 P50406 2/20 0.41
NMT1 P30419 1/20 0.40
HTR2A P28223 1/20 0.40
F10 P00742 1/20 0.39
BRD4 O60885 1/20 0.39
FFAR1 O14842 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7865968 0.90 CHRNB2 (0.42) CHRNB2CHRNA4PRMT5HTR6NMT1
SCHEMBL7863962 0.80 HTR2A (0.43) CHRNB2CHRNA4HTR2A
SCHEMBL7872529 0.80 REN (0.41) CHRNB2CHRNA4HTR2A
SCHEMBL10202520 0.78 REN (0.44) SLC6A2SLC6A4SLC6A3FFAR4PTGER1
SCHEMBL7863795 0.77 REN (0.54) HTR2A
SCHEMBL7863764 0.77 REN (0.58)
SCHEMBL7867634 0.76 REN (0.44) SLC6A2SLC6A4SLC6A3
SCHEMBL7870969 0.75 REN (0.49)
SCHEMBL7872769 0.75 REN (0.55)
SCHEMBL7875804 0.73 HTR2A (0.40) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed