SCHEMBL7875804

SCHEMBL7875804

COCc1ccc2cccc(-c3ccc([C@@H]4CCCNC4)c(C)c3)c2c1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.40
ACP1 P24666 1/20 0.38
IKBKB O14920 2/20 0.37
HTR2C P28335 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7872781 0.85 TLR8 (0.44) HTR2AIKBKB
SCHEMBL10202508 0.79 REN (0.38) HTR2A
SCHEMBL7863962 0.74 HTR2A (0.43) HTR2AHTR2C
SCHEMBL7867597 0.73 CHRNB2 (0.46) HTR2A
SCHEMBL7872529 0.69 REN (0.41) HTR2AIKBKB
SCHEMBL7863795 0.69 REN (0.54) HTR2AIKBKB
SCHEMBL7865968 0.68 CHRNB2 (0.42) IKBKB
SCHEMBL16446427 0.67 HTR2A (0.59) HTR2AIKBKBHTR2C
SCHEMBL7863764 0.67 REN (0.58) IKBKB
SCHEMBL26938735 0.67 HTR2A (0.54) HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed