SCHEMBL7868052

SCHEMBL7868052

COc1cc2c(C3=CCNCC3)c[nH]c2cc1F

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.62
ALDH1A1 P00352 3/20 0.62
HTR2C P28335 3/20 0.62
HSD17B10 Q99714 3/20 0.62
MAPT P10636 2/20 0.62
HTR6 P50406 2/20 0.62
MEN1 O00255 2/20 0.62
HTR1D P28221 2/20 0.62
KMT2A Q03164 2/20 0.62
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
MAPK1 P28482 1/20 0.62
BRCA1 P38398 1/20 0.62
DRD2 P14416 1/20 0.51
ALOX15 P16050 1/20 0.51
JAK2 O60674 1/20 0.49
PRKD3 O94806 1/20 0.49
MARK3 P27448 1/20 0.49
PRKCI P41743 1/20 0.49
PRKCD Q05655 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7867252 0.85 MAPT (0.62) KDM4EALDH1A1HTR2CHSD17B10MAPT
SCHEMBL16802081 0.78 HTR2C (0.55) KDM4EALDH1A1HTR2CHSD17B10MAPT
Ru-24969 SCHEMBL2359264 0.77 HTR6 (1.00) KDM4EALDH1A1HTR2CHSD17B10MAPT
SCHEMBL7864917 0.77 HTR6 (0.81) KDM4EALDH1A1HTR2CHSD17B10MAPT
Ru-24969 SCHEMBL29390076 0.77 HTR6 (1.00) KDM4EALDH1A1HTR2CHSD17B10MAPT
SCHEMBL7867382 0.77 CCNT1 (0.43) KDM4EALDH1A1HTR2CHSD17B10MAPT
SCHEMBL5845143 0.75 HTR2C (0.65) KDM4EALDH1A1HTR2CHSD17B10MAPT
SCHEMBL2778860 0.75 HTR6 (0.67) KDM4EALDH1A1HTR2CHSD17B10MAPT
SCHEMBL7866446 0.73 CCNT1 (0.49) CCNT1CDK9QDPR
Hydrochloric Acid SCHEMBL979625 0.72 QDPR (0.64) HTR2CCCNT1CDK9QDPRCD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed