Ru-24969

Ru-24969

SCHEMBL2359264

COc1ccc2[nH]cc(C3=CCNCC3)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 1.00
KDM4E B2RXH2 2/20 1.00
ALDH1A1 P00352 2/20 1.00
MAPT P10636 2/20 1.00
HTR2C P28335 2/20 1.00
HSD17B10 Q99714 2/20 1.00
MEN1 O00255 1/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
HTR1D P28221 1/20 1.00
MAPK1 P28482 1/20 1.00
BRCA1 P38398 1/20 1.00
KMT2A Q03164 1/20 1.00
JAK2 O60674 1/20 0.63
PRKD3 O94806 1/20 0.63
MARK3 P27448 1/20 0.63
PRKCI P41743 1/20 0.63
PRKCD Q05655 1/20 0.63
CAMK2B Q13554 1/20 0.63
CAMK2G Q13555 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ru-24969 SCHEMBL29390076 1.00 HTR6 (1.00) HTR6KDM4EALDH1A1MAPTHTR2C
Ru-24969 SCHEMBL29550112 0.90 HTR6 (0.81) HTR6KDM4EALDH1A1MAPTHTR2C
SCHEMBL7864917 0.90 HTR6 (0.81) HTR6KDM4EALDH1A1MAPTHTR2C
SCHEMBL6631651 0.82 KDM4E (0.70) HTR6KDM4EALDH1A1MAPTHTR2C
SCHEMBL8925573 0.82 HTR1D (0.69) HTR6KDM4EALDH1A1MAPTHTR2C
SCHEMBL5705100 0.80 KDM4E (0.66) HTR6KDM4EALDH1A1MAPTHTR2C
SCHEMBL7460028 0.80 HTR6 (0.67) HTR6KDM4EALDH1A1MAPTHTR2C
SCHEMBL3836149 0.80 HTR6 (0.67) HTR6KDM4EALDH1A1MAPTHTR2C
SCHEMBL1675799 0.80 HTR6 (0.67) HTR6KDM4EALDH1A1MAPTHTR2C
SCHEMBL2783986 0.80 HTR6 (0.67) HTR6KDM4EALDH1A1MAPTHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 120 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS INC (US) 2025-09-25 US claimed
WO-2023212244-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS, INC. (US) 2023-11-02 WO claimed
US-20220249440-A1 MUSCLE REGENERATION PROMOTER SATO PHARMACEUTICAL CO., LTD. (JP) 2022-08-11 US claimed
US-20140350064-A1 PHARMACEUTICAL COMPOSITION COMPRISING AN AMPK ACTIVATOR AND A SEROTONERGIC AGENT AND METHODS OF USE THEREOF ALS MOUNTAIN LLC 2014-11-27 US claimed
US-20120183600-A1 NOVEL COMPOSITION FOR TREATING METABOLIC SYNDROME AND OTHER CONDITIONS CHEN CHIEN-HUNG (US) 2012-07-19 US claimed
US-20050080084-A1 Compositions of a cyclooxygenase-2 selective inhibitor and a serotonin-modulating agent for the treatment of central nervous system damage PHARMACIA CORPORATION 2005-04-14 US claimed
EP-0455510-B1 Use of 5-HT1A receptor agonist compounds for inhibiting gastric acid secretion LILLY CO ELI (US) 1996-11-27 EP claimed
EP-0455510-A2 Use of 5-HT1A receptor agonist compounds for inhibiting gastric acid secretion ELI LILLY AND COMPANY (US) 1991-11-06 EP claimed
US-4196209-A Treating psychic disorders with piperidyl-indoles ROUSSEL UCLAF (FR) 1980-04-01 US claimed
JP-8027029-A None JP disclosed
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS INC (US) 2025-09-25 US disclosed
US-20250034106-A1 3-CYCLOAMINO-INDOLE COMPOUNDS AS SEROTONERGIC AGENTS USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO MINDSET PHARMA INC. (CA) 2025-01-30 US disclosed
US-20240376052-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS SEROTONERGIC AGENTS USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO MINDSET PHARMA INC. (CA) 2024-11-14 US disclosed
WO-2023212244-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS, INC. (US) 2023-11-02 WO disclosed
EP-0379314-A1 3-(1,2,5,6-Tetrahydropyridyl)-pyrrolopyridines PFIZER INC. (US) 1990-07-25 EP disclosed
EP-0360077-A2 Use of serotonin antagonists in the treatment of apoplexia cerebri Troponwerke GmbH & Co. KG (DE) 1990-03-28 EP disclosed
US-4855302-A 8-((4-(INDOL-3-YL)PIPERIDINO)ALKYL)-8-AZASPIRO(4.5)DECANE-7,9 -DIONES ROUSSEL UCLAF (FR) 1989-08-08 US disclosed
US-4278677-A Tetrahydropyridinyl indoles ROUSSEL UCLAF (FR) 1981-07-14 US disclosed
US-4232031-A Process for preparation of piperidyl-indoles ROUSSEL UCLAF (FR) 1980-11-04 US disclosed
US-4196209-A Treating psychic disorders with piperidyl-indoles ROUSSEL UCLAF (FR) 1980-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240376052-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS SEROTONERGIC AGENTS USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO TPH1, HTR5A, TPH2 HTR6 6/4885KDM4E 3293/4885ALDH1A1 1436/4885
US-20220249440-A1 MUSCLE REGENERATION PROMOTER MUSK, MYLK2, MYH2 HTR6 62/4885KDM4E 1326/4885ALDH1A1 1317/4885
US-20050080084-A1 Compositions of a cyclooxygenase-2 selective inhibitor and a serotonin-modulating agent for the treatment of central nervous system damage TPH2, TPH1, HTR2A HTR6 11/4885KDM4E 4399/4885ALDH1A1 1946/4885
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS HTR2A, HTR5A, HTR6 HTR6 3/4885KDM4E 4347/4885ALDH1A1 913/4885
US-20250034106-A1 3-CYCLOAMINO-INDOLE COMPOUNDS AS SEROTONERGIC AGENTS USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO TPH1, HTR3A, HTR1A HTR6 6/4885KDM4E 3948/4885ALDH1A1 1854/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.