Maleic Acid

Maleic Acid

SCHEMBL786851

NCCN.O=C(O)/C=C\C(=O)O.O=C(O)/C=C\C(=O)O

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.64
TP53 P04637 1/20 0.64
EGLN1 Q9GZT9 1/20 0.64
EGLN3 Q9H6Z9 1/20 0.64
KMT2A Q03164 2/20 0.59
MEN1 O00255 1/20 0.59
GABRR1 P24046 3/20 0.58
GABRR2 P28476 3/20 0.58
BLM P54132 3/20 0.58
GABRR3 A8MPY1 2/20 0.58
LMNA P02545 2/20 0.58
NPSR1 Q6W5P4 2/20 0.58
APEX1 P27695 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
HCAR2 Q8TDS4 6/20 0.44
GLRA1 P23415 1/20 0.41
SLC6A9 P48067 1/20 0.41
OR51E2 Q9H255 1/20 0.41
GABRP O00591 3/20 0.39
GABRD O14764 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL18065037 1.00 TSHR (0.64) TSHRTP53EGLN1EGLN3KMT2A
Fumaric Acid SCHEMBL2840791 1.00 TSHR (0.64) TSHRTP53EGLN1EGLN3KMT2A
Fumaric Acid SCHEMBL786567 1.00 TSHR (0.64) TSHRTP53EGLN1EGLN3KMT2A
Fumaric Acid SCHEMBL18065038 1.00 TSHR (0.64) TSHRTP53EGLN1EGLN3KMT2A
Maleic Acid SCHEMBL28320762 0.91 TSHR (0.53) TSHRTP53EGLN1EGLN3KMT2A
Ethylenediamine SCHEMBL28100956 0.88 TSHR (0.50) TSHRTP53EGLN1EGLN3KMT2A
Fumaric Acid SCHEMBL1835362 0.87 TSHR (0.56) TSHRTP53EGLN1EGLN3KMT2A
Maleic Acid SCHEMBL30550381 0.87 TSHR (0.56) TSHRTP53EGLN1EGLN3KMT2A
Maleic Acid SCHEMBL28650191 0.87 TSHR (0.56) TSHRTP53EGLN1EGLN3KMT2A
Fumaric Acid SCHEMBL8771350 0.87 TSHR (0.56) TSHRTP53EGLN1EGLN3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 140 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940228-B1 BAIT COMPOSITIONS COMPRISING AT LEAST ONE SPINOSYN AND ONE MOLLUSCICIDE NEUDORFF W GMBH KG (DE) 2015-07-29 EP claimed
US-20130206181-A1 AUTOMATIC DISHWASHING COMPOSITION INNOSPEC LIMITED (GB) 2013-08-15 US claimed
EP-2619301-A1 AUTOMATIC DISHWASHING COMPOSITION Innospec Limited (GB) 2013-07-31 EP claimed
WO-2012038755-A1 AUTOMATIC DISHWASHING COMPOSITION INNOSPEC LIMITED (GB) 2012-03-29 WO claimed
US-7964205-B2 Insecticide and molluscicide composition and methods W. NEUDORFF GMBH KG (DE) 2011-06-21 US claimed
EP-1940228-A2 BAIT COMPOSITIONS COMPRISING AT LEAST ONE SPINOSYN AND ONE MOLLUSCICIDE W. Neudorff GmbH KG (DE) 2008-07-09 EP claimed
US-20070148203-A1 Insecticide and molluscicide composition and methods W. NEUDORFF GMBH KG (DE) 2007-06-28 US claimed
WO-2007031565-A2 BAIT COMPOSITIONS COMPRISING AT LEAST ONE SPINOSYN AND ONE MOLLUSCICIDE W. NEUDORFF GMBH KG (DE) 2007-03-22 WO claimed
US-20030118625-A1 Ingestible molluscicide W. NEUDORFF GMBH KG (DE) 2003-06-26 US claimed
EP-1312260-A1 Ingestible molluscicide W. Neudorff GmbH KG (DE) 2003-05-21 EP claimed
EP-3891204-B1 POLYCARBOXYLIC ACID COMPOUNDS FOR THE TREATMENT OF FIBROUS AMINO ACID BASED SUBSTRATES, ESPECIALLY HAIR MOMENTIVE PERFORMANCE MAT INC (US) 2025-04-09 EP disclosed
EP-4396319-A1 MACHINE DISHWASH DETERGENT Unilever IP Holdings B.V. (NL) 2024-07-10 EP disclosed
EP-4396318-A1 MACHINE DISHWASH DETERGENT Unilever IP Holdings B.V. (NL) 2024-07-10 EP disclosed
EP-4396317-A1 MACHINE DISHWASH DETERGENT Unilever IP Holdings B.V. (NL) 2024-07-10 EP disclosed
US-20240218295-A1 MACHINE DISHWASH DETERGENT CONOPCO INC., D/B/A UNILEVER (US) 2024-07-04 US disclosed
US-6852329-B2 Transition metal compound and a complexing agent, and/or the complex of a transition metal compound and a complexing agents W. NEUDORFF GMBH KG (DE) 2005-02-08 US disclosed
US-20030118625-A1 Ingestible molluscicide W. NEUDORFF GMBH KG (DE) 2003-06-26 US disclosed
US-20030118625-A1 Ingestible molluscicide W. NEUDORFF GMBH KG (DE) 2003-06-26 US disclosed
EP-1312260-A1 Ingestible molluscicide W. Neudorff GmbH KG (DE) 2003-05-21 EP disclosed
EP-1312260-A1 Ingestible molluscicide W. Neudorff GmbH KG (DE) 2003-05-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030118625-A1 Ingestible molluscicide DDT, IDUA, NRDC TSHR 2221/4885TP53 4243/4885EGLN1 3932/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.