SCHEMBL7870752

SCHEMBL7870752

COc1cc2cc(C3=CCNCC3)sc2cc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QDPR P09417 1/20 0.42
ACHE P22303 1/20 0.40
CCNT1 O60563 11/20 0.39
CDK9 P50750 11/20 0.39
TLR9 Q9NR96 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
TGFBR1 P36897 1/20 0.36
ACVR1 Q04771 1/20 0.36
KCNH2 Q12809 1/20 0.36
CD274 Q9NZQ7 1/20 0.35
HTR6 P50406 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
HTR1D P28221 1/20 0.34
HTR2C P28335 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6312469 0.77 HTR6 (0.49) QDPRCCNT1CDK9HTR6KDM4E
SCHEMBL5758301 0.75 HTR6 (0.44) QDPRCCNT1CDK9HTR6HTR2C
SCHEMBL5756400 0.75 HTR6 (0.44) QDPRCCNT1CDK9HTR6HTR2C
SCHEMBL7867382 0.74 CCNT1 (0.43) QDPRCCNT1CDK9TLR9TLR7
SCHEMBL7866446 0.73 CCNT1 (0.49) QDPRCCNT1CDK9
SCHEMBL16874849 0.70 QDPR (0.66) QDPRCCNT1CDK9TLR9TLR7
SCHEMBL27553177 0.70 QDPR (0.70) QDPRCCNT1CDK9TLR9TLR7
SCHEMBL4359750 0.70 SIGMAR1 (0.50) QDPRKDM4EALDH1A1MAPTHTR2C
Hydrochloric Acid SCHEMBL979625 0.69 QDPR (0.64) QDPRCCNT1CDK9TLR9TLR7
SCHEMBL7867931 0.69 HTR2C (0.41) CCNT1CDK9HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
WO-1997047302-A1 INHIBITION OF SEROTONIN REUPTAKE ELI LILLY AND COMPANY (US) 1997-12-18 WO disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed