SCHEMBL7871377

SCHEMBL7871377

CC(=N)Nc1ccc2cn[nH]c2c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 13/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2D6 P10635 1/20 0.67
CYP2C9 P11712 1/20 0.67
CYP2C19 P33261 1/20 0.67
HIF1A Q16665 1/20 0.67
PHLPP2 Q6ZVD8 1/20 0.67
HSD17B10 Q99714 1/20 0.67
MAPT P10636 12/20 0.61
KDM4E B2RXH2 10/20 0.61
HPGD P15428 2/20 0.59
GAA P10253 2/20 0.58
RAB9A P51151 1/20 0.58
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
F2 P00734 2/20 0.57
HTT P42858 2/20 0.57
ROCK2 O75116 1/20 0.55
ROCK1 Q13464 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14045319 0.84 ROCK2 (0.77) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL27692289 0.83 ALDH1A1 (0.61) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL24797472 0.80 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1548213 0.79 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL30725947 0.79 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4194552 0.78 ALDH1A1 (0.62) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8774349 0.77 ALDH1A1 (0.67) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL30026503 0.77 ALDH1A1 (0.67) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5823003 0.77 ALDH1A1 (0.77) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL22590423 0.77 ALDH1A1 (0.61) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37438-E1 Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase GLAXO WELLCOME INC. 2001-11-06 US disclosed
US-5866612-A Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase GLAXO WELLCOME INC. (US) 1999-02-02 US disclosed
EP-0799191-A1 ACETAMIDINE DERIVATIVES AND THEIR USE AS INHIBITORS FOR THE NITRIC OXIDE SYNTHASE THE WELLCOME FOUNDATION LIMITED (GB) 1997-10-08 EP disclosed
WO-1996019440-A1 ACETAMIDINE DERIVATIVES AND THEIR USE AS INHIBITORS FOR THE NITRIC OXIDE SYNTHASE THE WELLCOME FOUNDATION LIMITED (GB) 1996-06-27 WO disclosed