SCHEMBL7864235

SCHEMBL7864235

CCCCCC1C(C(=O)OCC#Cc2cccnc2)=C(C)NC(c2cccc(-n3ccnc3)c2)=C1C(=O)OCC

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.38
TRPV1 Q8NER1 1/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.37
CACNA1C Q13936 3/20 0.36
TMIGD3 P0DMS9 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GAA P10253 1/20 0.34
CYP3A4 P08684 2/20 0.34
GRM5 P41594 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7869546 0.91 ADORA3 (0.41) ADORA3TRPV1MAPTMAPK1CACNA1C
SCHEMBL7871519 0.88 ADORA3 (0.37) ADORA3TRPV1MAPTMAPK1TMIGD3
SCHEMBL7872517 0.86 ADORA3 (0.38) ADORA3TRPV1MAPTMAPK1CACNA1C
SCHEMBL8324841 0.85 ADORA3 (0.46) ADORA3TRPV1MAPTMAPK1CACNA1C
SCHEMBL7876066 0.84 ADORA3 (0.36) ADORA3MAPTMAPK1CACNA1CTMIGD3
SCHEMBL7871558 0.83 ADORA3 (0.43) ADORA3TRPV1MAPTMAPK1CACNA1C
SCHEMBL7869557 0.80 ADORA3 (0.42) ADORA3TRPV1MAPTMAPK1CACNA1C
SCHEMBL7876069 0.79 ADORA3 (0.39) ADORA3TRPV1MAPK1TMIGD3NPSR1
SCHEMBL7871376 0.78 ADORA3 (0.37) ADORA3TRPV1MAPTMAPK1TMIGD3
SCHEMBL7873250 0.78 ADORA3 (0.37) ADORA3TRPV1MAPTMAPK1TMIGD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed