SCHEMBL7872416

SCHEMBL7872416

CC(=O)N1CCN(C(=O)c2ccc(C)cc2F)CC1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CPS1 P31327 6/20 0.57
HTT P42858 4/20 0.54
TSHR P16473 3/20 0.54
LMNA P02545 2/20 0.54
MAPT P10636 1/20 0.54
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HSP90AA1 P07900 1/20 0.47
HPGD P15428 1/20 0.45
TP53 P04637 1/20 0.44
EPHX2 P34913 1/20 0.43
PDE2A O00408 1/20 0.43
MEN1 O00255 1/20 0.43
MAPK1 P28482 1/20 0.43
GFER P55789 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18010744 0.88 CPS1 (0.57) CPS1HTTTSHRLMNAMAPT
SCHEMBL7878686 0.87 CPS1 (0.60) CPS1HTTTSHRLMNAMAPT
SCHEMBL12205464 0.86 CPS1 (0.58) CPS1HTTTSHRLMNAMAPT
SCHEMBL24910640 0.84 LMNA (0.53) HTTTSHRLMNAMAPTKDM4E
SCHEMBL7878481 0.84 ALDH1A1 (0.55) CPS1HTTTSHRLMNAMAPT
SCHEMBL7870107 0.84 CPS1 (0.54) CPS1HTTTSHRLMNAMAPT
SCHEMBL17400772 0.83 CPS1 (0.56) CPS1HTTTSHRLMNAMAPT
SCHEMBL7878741 0.83 CPS1 (0.52) CPS1HTTTSHRLMNAMAPT
SCHEMBL7872429 0.83 MAPT (0.57) CPS1HTTTSHRLMNAMAPT
SCHEMBL7870100 0.82 CPS1 (0.59) CPS1HTTTSHRLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010122069-A1 5-ALKYNYL-PYRIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-10-28 WO disclosed