SCHEMBL7872469

SCHEMBL7872469

CC(CNc1ncc[nH]c1=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.41
AOC3 Q16853 1/20 0.41
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
KAT2B Q92831 5/20 0.37
BCHE P06276 1/20 0.36
DAO P14920 1/20 0.36
JAK3 P52333 2/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4158770 0.72 MEN1 (0.51) TAAR1KMT2AJAK2JAK1
SCHEMBL13939838 0.70 GPR84 (0.47)
SCHEMBL3647566 0.70 HTT (0.40) TAAR1AOC3KMT2A
SCHEMBL6647148 0.69 JAK2 (0.40) JAK2JAK1
SCHEMBL22524173 0.69 LMNA (0.44) TAAR1AOC3KMT2APOLB
SCHEMBL3773150 0.68 TAAR1 (0.53) TAAR1HRH4
SCHEMBL1522424 0.67 HTT (0.60) KMT2AJAK3JAK2JAK1
SCHEMBL7878663 0.67 NISCH (0.43) TAAR1DAO
SCHEMBL10569996 0.66 ALDH1A1 (0.38) KMT2A
SCHEMBL11393997 0.66 TAAR1 (0.52) TAAR1AOC3KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086122-A1 PYRAZINONE PROTEASE INHIBITORS Johnson & Johnson Pharmaceutical Research & Development, L.L.C. (US) 2001-03-28 EP claimed
WO-1999064446-A1 PYRAZINONE PROTEASE INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1999-12-16 WO claimed