SCHEMBL7874969

SCHEMBL7874969

CC(=N)Nc1cccc(CNCc2cccc(NC(C)=N)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.46
NOS3 P29474 2/20 0.43
NOS2 P35228 2/20 0.43
MAPT P10636 2/20 0.40
SLC2A4 P14672 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CHRM2 P08172 2/20 0.39
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7875011 0.88 NOS1 (0.49) NOS1NOS3NOS2MAPTNPSR1
SCHEMBL7873162 0.88 NOS1 (0.49) NOS1NOS2MAPTNPSR1GRIN2D
SCHEMBL7874966 0.86 CYP3A4 (0.51) NOS1NOS3NOS2MAPTNPSR1
SCHEMBL14367988 0.84 SIGMAR1 (0.54) MAPTMEN1KMT2AGRIN2DGRIN3B
SCHEMBL7865754 0.84 PDK1 (0.51) MAPTNPSR1GRIN2DGRIN3BGRIN1
SCHEMBL5080879 0.82 LOXL2 (0.49) NOS1NOS3NOS2GRIN2DGRIN3B
Hydrochloric Acid SCHEMBL7875006 0.81 LOXL2 (0.47) NOS1NOS3NOS2GRIN2DGRIN3B
SCHEMBL7873185 0.81 TRPV1 (0.46) MAPTNPSR1GRIN2DGRIN3BGRIN1
SCHEMBL7865767 0.80 POLB (0.47) MAPTMEN1KMT2ACYP1A2RAB9A
SCHEMBL5078291 0.79 NOS1 (0.49) NOS1NOS3NOS2GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37438-E1 Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase GLAXO WELLCOME INC. 2001-11-06 US disclosed
US-5866612-A Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase GLAXO WELLCOME INC. (US) 1999-02-02 US disclosed