SCHEMBL7877237

SCHEMBL7877237

C=C(c1nccs1)N1CCN(C2CNC2)CC1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 17/20 0.36
MITF O75030 1/20 0.34
HSP90AA1 P07900 1/20 0.34
FAAH O00519 1/20 0.34
HKDC1 Q2TB90 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL693819 0.83 MGLL (0.50) MGLLFAAH
Hydrochloric Acid SCHEMBL14813360 0.82 MGLL (0.49) MGLLFAAH
SCHEMBL7723818 0.74 ALDH1A1 (0.38) MGLLALDH1A1
SCHEMBL13148464 0.73 MGLL (0.51) MGLLFAAH
SCHEMBL8379841 0.72 ALDH1A1 (0.41) MGLLMITFHSP90AA1HKDC1ALDH1A1
SCHEMBL16862126 0.69 MGLL (0.52) MGLLFAAH
SCHEMBL30359147 0.67 ALDH1A1 (0.42) MGLLHKDC1ALDH1A1
SCHEMBL2721136 0.64 RBP4 (0.51) MGLLALDH1A1
SCHEMBL584468 0.64 CHRNA4 (0.55)
SCHEMBL16862045 0.62 MGLL (0.51) MGLLFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010124082-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-10-28 WO disclosed
WO-2010124114-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-10-28 WO disclosed
WO-2010124108-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-10-28 WO disclosed
WO-2010124102-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-10-28 WO disclosed
WO-2010124119-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-10-28 WO disclosed
WO-2010124112-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-10-28 WO disclosed
WO-2010124086-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-10-28 WO disclosed
WO-2010124116-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2010-10-28 WO disclosed