SCHEMBL30359147

SCHEMBL30359147

O=C(c1nccs1)N1C2CCC1CNC2

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
RBP4 P02753 1/20 0.40
RBBP9 O75884 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36
SMO Q99835 1/20 0.34
GRM5 P41594 3/20 0.34
MGLL Q99685 6/20 0.34
TNKS O95271 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
MAPT P10636 1/20 0.33
HKDC1 Q2TB90 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL693819 0.78 MGLL (0.50) RBP4SMOMGLL
Hydrochloric Acid SCHEMBL14813360 0.77 MGLL (0.49) RBP4SMOMGLL
SCHEMBL584468 0.76 CHRNA4 (0.55)
SCHEMBL2721136 0.75 RBP4 (0.51) ALDH1A1RBP4SMOMGLL
SCHEMBL30359120 0.75 TRPV4 (0.42) ALDH1A1TRPV4
SCHEMBL7723818 0.74 ALDH1A1 (0.38) ALDH1A1RBP4RBBP9MGLL
SCHEMBL30359028 0.74 TRPV4 (0.41) ALDH1A1TRPV4MGLL
SCHEMBL584771 0.74 CHRNA4 (0.57)
SCHEMBL2130529 0.71 CYP3A4 (0.46) ALDH1A1RBP4SMOMGLLHKDC1
SCHEMBL2130521 0.71 CYP3A4 (0.46) ALDH1A1RBP4SMOMGLLHKDC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057057-A Conjugates of alpha 2-adrenoceptor subtype C (alpha-2C) antagonists and TASK1/3 channel blockers for the treatment of sleep apnea 拜耳公司 2023-05-02 CN disclosed