SCHEMBL7877508

SCHEMBL7877508

CN1CCN(c2ccccc2CCNC(=O)c2ncc(-c3ccccc3)o2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 14/20 0.50
HDAC1 Q13547 13/20 0.50
HDAC3 O15379 2/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
USP30 Q70CQ3 1/20 0.47
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43
TUBA1A Q71U36 1/20 0.43
TUBA1C Q9BQE3 1/20 0.43
TUBB6 Q9BUF5 1/20 0.43
TUBB2B Q9BVA1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28611017 0.79 HIF1A (0.61) HDAC6HDAC1HDAC3HDAC2HDAC8
SCHEMBL5160839 0.79 DRD2 (0.53) POLBMAPK1
SCHEMBL7871309 0.75 DRD2 (0.56) HDAC1SNCA
SCHEMBL5160692 0.75 HTR1A (0.59)
SCHEMBL19017785 0.73 USP30 (0.74) HDAC6HDAC1HDAC3HDAC2HDAC8
SCHEMBL6662366 0.73 NPC1 (0.52)
SCHEMBL5160955 0.73 HTR1A (0.60) MAPK1
SCHEMBL28610666 0.72 HIF1A (0.65) HDAC6HDAC1HDAC3HDAC2HDAC8
SCHEMBL24089868 0.72 HDAC6 (0.62) HDAC6HDAC1HDAC3HDAC2HDAC8
SCHEMBL7875925 0.71 DRD2 (0.54) SNCAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020183011-A1 HTR1D INHIBITORS AND USES THEREOF IN THE TREATMENT OF CANCER INSTITUT CURIE (FR) 2020-09-17 WO disclosed
US-6323229-B1 COMPOUNDS ARE USEFUL PSYCHOTHERAPEUTICS AND ARE POTENT AGONISTS AND/OR ANTAGONISTS OF THE SEROTONIN 1A (5-HT 1A) AND/OR SEROTONIN 1D (5-HT 1D) FOR TREATMENT OF HYPERTENSION, DEPRESSION, GENERALIZED ANXIETY DISORDER PFIZER INC 2001-11-27 US disclosed
US-6197773-B1 HEADACHES; ANTIDEPRESSANTS PFIZER INC 2001-03-06 US disclosed