SCHEMBL7871309

SCHEMBL7871309

CN1CCN(c2ccccc2CCNC(=O)c2ccc(-c3ccccc3)s2)CC1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.56
DRD4 P21917 2/20 0.56
DRD3 P35462 2/20 0.56
ACKR3 P25106 14/20 0.53
KDM4E B2RXH2 1/20 0.46
NPC1 O15118 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
SNCA P37840 1/20 0.46
HDAC1 Q13547 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7875925 0.86 DRD2 (0.54) DRD2DRD4DRD3NPC1ALDH1A1
SCHEMBL5160839 0.81 DRD2 (0.53) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL6662366 0.77 NPC1 (0.52) DRD2DRD4DRD3KDM4ENPC1
SCHEMBL7158123 0.76 AKT3 (0.52) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL5160692 0.75 HTR1A (0.59) RAB9A
SCHEMBL5160955 0.75 HTR1A (0.60) DRD2DRD4DRD3KDM4ENPC1
SCHEMBL7877508 0.75 HDAC6 (0.50) SNCAHDAC1
SCHEMBL7160985 0.74 ESRRG (0.52) DRD2DRD4DRD3ACKR3ALDH1A1
SCHEMBL6660894 0.73 HCN1 (0.53) DRD2DRD4DRD3KDM4ENPC1
Hydrochloric Acid SCHEMBL7154175 0.73 ESRRG (0.50) DRD2DRD4DRD3ACKR3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020183011-A1 HTR1D INHIBITORS AND USES THEREOF IN THE TREATMENT OF CANCER INSTITUT CURIE (FR) 2020-09-17 WO disclosed
US-6323229-B1 COMPOUNDS ARE USEFUL PSYCHOTHERAPEUTICS AND ARE POTENT AGONISTS AND/OR ANTAGONISTS OF THE SEROTONIN 1A (5-HT 1A) AND/OR SEROTONIN 1D (5-HT 1D) FOR TREATMENT OF HYPERTENSION, DEPRESSION, GENERALIZED ANXIETY DISORDER PFIZER INC 2001-11-27 US disclosed
US-6197773-B1 HEADACHES; ANTIDEPRESSANTS PFIZER INC 2001-03-06 US disclosed