SCHEMBL7877903

SCHEMBL7877903

C=CCOC(=O)CNC(=O)C(NC(=O)[C@H](CC(=O)OC(C)(C)C)NC(=O)OCc1ccccc1)c1ccc(OC(C)(C)C)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.46
CTSK P43235 1/20 0.46
CTSS P25774 2/20 0.44
ABCB1 P08183 1/20 0.43
CASP3 P42574 4/20 0.41
CASP7 P55210 4/20 0.41
CASP1 P29466 4/20 0.41
CASP4 P49662 2/20 0.41
SYK P43405 1/20 0.41
CASP9 P55211 2/20 0.40
CASP10 Q92851 2/20 0.40
CASP8 Q14790 1/20 0.40
CTSB P07858 1/20 0.40
MMP8 P22894 1/20 0.40
MAPT P10636 1/20 0.39
BACE1 P56817 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7878944 0.87 CTSL (0.52) CTSLCTSKCTSSCASP3CASP7
SCHEMBL7885844 0.82 CASP3 (0.54) CTSLCTSKCTSSCASP3CASP7
SCHEMBL7888466 0.82 CASP3 (0.52) CTSLCTSKCTSSCASP3CASP7
SCHEMBL19015914 0.82 CASP3 (0.52) CTSLCTSKCTSSCASP3CASP7
SCHEMBL19015807 0.81 CTSL (0.53) CTSLCTSKCTSSCTSB
SCHEMBL7971579 0.81 CTSL (0.51) CTSLCTSKABCB1CASP3CASP7
SCHEMBL7888201 0.80 CTSL (0.52) CTSLCTSKCTSSCTSB
SCHEMBL7888191 0.79 CTSK (0.53) CTSLCTSKCTSSCASP3CASP1
SCHEMBL7886440 0.79 CTSK (0.52) CTSLCTSKCTSSCASP3CASP7
SCHEMBL7886897 0.78 CTSK (0.44) CTSLCTSKCTSSCASP3SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010133000-A1 SELECTIVE CASPASE INHIBITORS AND USES THEREOF NEW WORLD LABORATORIES INC. (CA) 2010-11-25 WO disclosed