SCHEMBL7888191

SCHEMBL7888191

C=CCOC(=O)CNC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)[C@H](CC(=O)OC(C)(C)C)NC(=O)OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.53
CTSS P25774 3/20 0.53
CASP3 P42574 2/20 0.51
CASP1 P29466 5/20 0.46
REN P00797 1/20 0.44
TGM2 P21980 1/20 0.43
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
CTSB P07858 3/20 0.42
CTSL P07711 3/20 0.42
NMBR P28336 2/20 0.42
PSMB1 P20618 1/20 0.42
PSMB8 P28062 1/20 0.42
PSMB9 P28065 1/20 0.42
PSMB5 P28074 1/20 0.42
PSMB10 P40306 1/20 0.42
PSMB2 P49721 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9962153 0.90 CASP3 (0.59) CTSKCTSSCASP3CASP1REN
SCHEMBL9961959 0.83 CASP3 (0.62) CTSKCTSSCASP3CASP1REN
SCHEMBL7888622 0.82 CASP3 (0.53) CTSKCTSSCASP3CASP1REN
SCHEMBL29358005 0.81 CASP3 (0.50) CTSKCTSSCASP3CASP1REN
SCHEMBL19944839 0.80 NMBR (0.59) CTSKCTSSCASP3CASP1REN
SCHEMBL9962288 0.80 CASP3 (0.60) CTSKCASP3CASP1RENCTSB
SCHEMBL19015914 0.80 CASP3 (0.52) CTSKCTSSCASP3CASP1TGM2
SCHEMBL7888466 0.80 CASP3 (0.52) CTSKCTSSCASP3CASP1TGM2
SCHEMBL7877903 0.79 CTSL (0.46) CTSKCTSSCASP3CASP1MAPT
SCHEMBL19606065 0.78 CASP1 (0.58) CTSKCTSSCASP3CASP1REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010133000-A1 SELECTIVE CASPASE INHIBITORS AND USES THEREOF NEW WORLD LABORATORIES INC. (CA) 2010-11-25 WO disclosed