SCHEMBL7878035

SCHEMBL7878035

Bc1cnc(N(C(C)=O)C(C)=O)c(COC(C)=O)c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 2/20 0.32
HSD17B10 Q99714 2/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12985694 0.83 CYP3A4 (0.35) CYP3A4ALDH1A1KDM4EHSD17B10HTT
SCHEMBL2067654 0.75 DGAT1 (0.37) CYP3A4
SCHEMBL7871957 0.68 DPP4 (0.36) ALDH1A1
SCHEMBL3293016 0.66 ALDH1A1 (0.52) CYP3A4ALDH1A1KDM4EHSD17B10
SCHEMBL11015127 0.64 SMN1; SMN2 (0.39) CYP3A4ALDH1A1KDM4EHSD17B10
SCHEMBL4074495 0.63 HSD17B10 (0.40) CYP3A4ALDH1A1KDM4EHSD17B10
SCHEMBL9013438 0.62 ALDH1A1 (0.37) CYP3A4ALDH1A1KDM4EHSD17B10
SCHEMBL12069180 0.62 MAOB (0.42) CYP3A4ALDH1A1KDM4EHSD17B10
SCHEMBL11013415 0.61 SMN1; SMN2 (0.37) CYP3A4ALDH1A1KDM4EHSD17B10
SCHEMBL11011350 0.61 SMN1; SMN2 (0.37) CYP3A4ALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139747-A1 1H-IMIDAZO[4, 5-c]QUINOLINONE COMPOUNDS, USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES NOVARTIS AG (CH) 2010-12-09 WO disclosed