SCHEMBL7879334

SCHEMBL7879334

CC(C)(C)Cn1nnc2c(Br)c(NCc3ccc(N)c(F)c3)ccc21

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 4/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
PIM1 P11309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7884054 0.82 ADRA2B (0.40) GRM2ADORA3ADORA2AADORA2BADORA1
SCHEMBL7875245 0.81 GRM2 (0.40) GRM2PIM1
SCHEMBL7879169 0.81 CCNB2 (0.36) GRM2ADORA3ADORA2AADORA2BADORA1
SCHEMBL7876318 0.80 GRM2 (0.31) GRM2
SCHEMBL7886812 0.80 TDO2 (0.40)
SCHEMBL7882339 0.80 MAPT (0.35) GRM2
SCHEMBL7884632 0.78 NMT1 (0.37) ADORA3ADORA2AADORA2BADORA1PIM1
SCHEMBL7879380 0.78 P2RX7 (0.36) GRM2
SCHEMBL7882812 0.78 GRM2 (0.40) GRM2
SCHEMBL7882669 0.78 RORC (0.38) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114726-A1 AMINOBENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed