SCHEMBL7880296

SCHEMBL7880296

COC(=O)c1ccc2c(CCCCN3CCCC(Cc4ccc(C#N)cc4)C3)c[nH]c2c1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 11/20 0.48
NPC1 O15118 1/20 0.46
SLC6A4 P31645 2/20 0.44
ACHE P22303 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7881273 0.94 HTR1A (0.53) HTR1ASLC6A4ACHESLC6A2SLC6A3
SCHEMBL7877114 0.91 NPC1 (0.49) HTR1ANPC1SLC6A4ACHE
SCHEMBL7878911 0.90 CCR3 (0.49) HTR1ANPC1
SCHEMBL7879009 0.90 HTR1A (0.55) HTR1ANPC1SLC6A4
SCHEMBL7075871 0.89 HTR1A (0.43) HTR1A
SCHEMBL7879034 0.85 HTR1A (0.55) HTR1ASLC6A4
SCHEMBL7082018 0.84 HTR1A (0.48) HTR1A
SCHEMBL7880274 0.84 HTR1A (0.55) HTR1ASLC6A4ACHE
SCHEMBL7880351 0.83 HTR1A (0.54) HTR1ASLC6A4
SCHEMBL7881308 0.83 ADRA2A (0.58) HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed