SCHEMBL7879009

SCHEMBL7879009

COC(=O)c1ccc2c(CCCCN3CCCC(Cc4ccccc4)C3)c[nH]c2c1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.55
NPC1 O15118 1/20 0.50
HTR2A P28223 1/20 0.48
CCR3 P51677 1/20 0.48
CHRNB2 P17787 2/20 0.48
CHRNB4 P30926 2/20 0.48
CHRNA3 P32297 2/20 0.48
CHRNA4 P43681 2/20 0.48
SLC6A4 P31645 2/20 0.47
CARM1 Q86X55 1/20 0.46
PRMT6 Q96LA8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959565 0.93 HTR1A (0.63) HTR1ASLC6A4
SCHEMBL7877114 0.93 NPC1 (0.49) HTR1ANPC1HTR2ACCR3SLC6A4
SCHEMBL7878911 0.92 CCR3 (0.49) HTR1ANPC1HTR2ACCR3
SCHEMBL7880296 0.90 HTR1A (0.48) HTR1ANPC1SLC6A4
SCHEMBL6955648 0.88 HTR2A (0.48) HTR1AHTR2ACCR3CHRNB2CHRNB4
SCHEMBL7879034 0.87 HTR1A (0.55) HTR1ASLC6A4
SCHEMBL6947219 0.86 HTR1A (0.52) HTR1AHTR2ACCR3SLC6A4
SCHEMBL7880274 0.86 HTR1A (0.55) HTR1ASLC6A4
SCHEMBL7881308 0.85 ADRA2A (0.58) HTR1ASLC6A4
SCHEMBL7880351 0.85 HTR1A (0.54) HTR1AHTR2ACCR3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed