SCHEMBL78865

SCHEMBL78865

COCCCn1cc(C(C)(C)C)c2cc(F)ccc21

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ICMT O60725 4/20 0.42
GSK3B P49841 2/20 0.39
CNR1 P21554 2/20 0.39
CNR2 P34972 2/20 0.39
HTR6 P50406 2/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
IDO1 P14902 1/20 0.35
CHUK O15111 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HTR3A P46098 3/20 0.35
LMNA P02545 2/20 0.34
MAPK1 P28482 2/20 0.34
HTT P42858 2/20 0.34
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78476 0.90 ICMT (0.42) ICMTGSK3BCNR1CNR2HTR6
SCHEMBL4602810 0.82 ICMT (0.44) ICMTGSK3BCNR1CNR2HTR6
SCHEMBL4602804 0.81 ICMT (0.43) ICMTGSK3BCNR1CNR2HTR6
SCHEMBL78417 0.81 CNR2 (0.53) CNR1CNR2ALDH1A1LMNAMAPK1
SCHEMBL91289 0.80 ICMT (0.55) ICMTGSK3BCNR1CNR2KDM4E
SCHEMBL13131421 0.79 MAP3K14 (0.35) ICMTGSK3BCNR1CNR2ALDH1A1
SCHEMBL8241203 0.78 ALDH1A1 (0.58) KDM4EALDH1A1LMNAHTTMAPT
SCHEMBL25403772 0.77 CNR1 (0.50) ICMTCNR1CNR2KDM4EALDH1A1
SCHEMBL31083818 0.77 CNR1 (0.50) ICMTCNR1CNR2KDM4EALDH1A1
SCHEMBL30564140 0.77 SMN1; SMN2 (0.56) ICMTCNR1CNR2ALDH1A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed