SCHEMBL78476

SCHEMBL78476

COCCCn1cc(C(C)(C)C)c2ccc(F)cc21

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ICMT O60725 3/20 0.42
HTR6 P50406 1/20 0.40
CNR1 P21554 5/20 0.37
CNR2 P34972 5/20 0.37
HRH2 P25021 3/20 0.37
CHUK O15111 1/20 0.35
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
PER2 O15055 1/20 0.33
CRY1 Q16526 1/20 0.33
CRY2 Q49AN0 1/20 0.33
GSK3B P49841 1/20 0.33
IL1B P01584 1/20 0.33
P2RX7 Q99572 1/20 0.33
MAP3K14 Q99558 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78865 0.90 ICMT (0.42) ICMTHTR6CNR1CNR2CHUK
SCHEMBL4602445 0.82 ICMT (0.44) ICMTHTR6CNR1CNR2HRH2
SCHEMBL4602440 0.81 ICMT (0.43) ICMTHTR6CNR1CNR2HRH2
SCHEMBL78417 0.81 CNR2 (0.53) CNR1CNR2LMNAMAPK1HTT
SCHEMBL91271 0.80 ICMT (0.54) ICMTHTR6CNR1CNR2HRH2
SCHEMBL13131421 0.79 MAP3K14 (0.35) ICMTCNR1CNR2CHUKLMNA
SCHEMBL8247540 0.78 ALDH1A1 (0.55) ICMTCNR1CNR2HRH2LMNA
SCHEMBL91362 0.76 REN (0.43) CNR1CNR2LMNAHTTGSK3B
SCHEMBL4602810 0.74 ICMT (0.44) ICMTHTR6CNR1CNR2LMNA
SCHEMBL22316061 0.74 SCN9A (0.44) ICMTHTR6CNR2GSK3BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed