SCHEMBL7887985

SCHEMBL7887985

[CH](CCCN1CCOCC1)C1CCNCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HRH3 Q9Y5N1 1/20 0.37
GNAO1 P09471 5/20 0.36
GNAI3 P08754 4/20 0.36
GNAI1 P63096 4/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 1/20 0.36
DUSP3 P51452 1/20 0.36
POLB P06746 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
LMNA P02545 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
EPHX1 P07099 1/20 0.34
GAA P10253 1/20 0.34
MAPK1 P28482 1/20 0.33
HIF1A Q16665 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7119085 0.90 KDM4E (0.36) KEAP1SMN1; SMN2HRH3GNAO1GNAI3
SCHEMBL7119089 0.75 GNAO1 (0.51) KEAP1SMN1; SMN2HRH3GNAO1GNAI3
SCHEMBL6408637 0.74 KEAP1 (0.58) KEAP1SMN1; SMN2HRH3CYP1A2HPGD
SCHEMBL5848078 0.74 CXCR4 (0.37) SMN1; SMN2HRH3GNAO1GNAI3GNAI1
SCHEMBL7887988 0.73 GNAO1 (0.54) KEAP1SMN1; SMN2HRH3GNAO1GNAI3
SCHEMBL3950022 0.73 SLC6A2 (0.31) HRH3
SCHEMBL6674597 0.73 SMN1; SMN2 (0.56) KEAP1SMN1; SMN2HRH3HPGDDUSP3
SCHEMBL151418 0.73 CXCR4 (0.57) KEAP1SMN1; SMN2HRH3CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL8901169 0.72 GNAO1 (0.56) KEAP1SMN1; SMN2HRH3GNAO1GNAI3
SCHEMBL15173760 0.71 KEAP1 (0.54) KEAP1SMN1; SMN2HRH3CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1119567-A1 QUINAZOLINE DERIVATIVES AstraZeneca AB (SE) 2001-08-01 EP disclosed
WO-2000021955-A1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2000-04-20 WO disclosed