SCHEMBL7888367

SCHEMBL7888367

Cc1cc(OC(=O)NCc2cccc([N+](=O)[O-])c2)c(N)s1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.47
PTPN1 P18031 3/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
MAPT P10636 2/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP2C19 P33261 2/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
RECQL P46063 1/20 0.44
AKR1B1 P15121 2/20 0.43
OPRM1 P35372 1/20 0.43
OPRK1 P41145 1/20 0.43
SETD7 Q8WTS6 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7890873 0.88 PTPN1 (0.47) ACKR3PTPN1MEN1KMT2AMAPT
SCHEMBL7886936 0.87 PTPN1 (0.48) ACKR3PTPN1MEN1KMT2AMAPT
SCHEMBL7880879 0.83 NCEH1 (0.48) ALDH1A1CYP2C19CYP2D6CYP2C9CYP1A2
SCHEMBL8211512 0.81 ACKR3 (0.55) ACKR3PTPN1MEN1KMT2AMAPT
SCHEMBL7893101 0.79 ALDH1A1 (0.56) MEN1KMT2AMAPTALDH1A1CYP2C19
SCHEMBL7889273 0.76 FAAH (0.48) KMT2AMAPTALDH1A1
SCHEMBL7426581 0.76 TSHR (0.49) MEN1KMT2AALDH1A1
SCHEMBL3275588 0.76 ACKR3 (0.59) ACKR3PTPN1MEN1KMT2AALDH1A1
SCHEMBL7890923 0.75 PTPN1 (0.44) ACKR3PTPN1MEN1KMT2AMAPT
SCHEMBL4582840 0.73 PTPN1 (0.63) ACKR3PTPN1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934301-B1 AMINOTHIOPHENE CARBOXYLIC ACID AMIDES AND THE USE THEREOF AS PHOSPHODIESTERASE INHIBITORS MERCK PATENT GMBH (DE) 2001-06-20 EP disclosed