SCHEMBL7894809

SCHEMBL7894809

N#Cc1c(O)ccnc1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNMA1 Q12791 1/20 0.38
ALDH1A1 P00352 7/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
KDM4E B2RXH2 4/20 0.37
GAA P10253 2/20 0.37
MAPT P10636 1/20 0.37
CACNA1B Q00975 1/20 0.37
APBA1 Q02410 1/20 0.37
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4C Q9H3R0 1/20 0.32
CA12 O43570 1/20 0.31
CA2 P00918 1/20 0.31
CA3 P07451 1/20 0.31
CA6 P23280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657787 0.78 KCNMA1 (0.36) KCNMA1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL6569026 0.78 ALDH1A1 (0.41) KCNMA1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL15741203 0.78 LRRK2 (0.40) KCNMA1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL31437529 0.78 KCNMA1 (0.36) KCNMA1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL5802874 0.78 KCNMA1 (0.40) KCNMA1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL28432011 0.78 EGLN2 (0.36) KCNMA1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL8242638 0.74 ALDH1A1 (0.53) KCNMA1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL15748249 0.74 MEN1 (0.35) KCNMA1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL172315 0.74 ALDH1A1 (0.53) ALDH1A1MEN1KMT2AKDM4EGAA
SCHEMBL29381656 0.72 ALDH1A1 (0.48) KCNMA1ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922543-B1 SUBSTITUTED PYRIDONE DERIVATIVES AS PDE10 INHIBITORS MERCK SHARP & DOHME (US) 2017-05-24 EP disclosed
US-6197964-B1 CHLORINATION USING BASIC CATALYST; DESALTING, HYDROLYSIS BAYER AKTIENGESELLSCHAFT (DE) 2001-03-06 US disclosed
EP-0973745-A1 METHOD FOR THE PRODUCTION OF 2,6-DICHLORO-5-FLUORONICOTINONITRILE AND THE CHEMICAL COMPOUND 3-CYANO-2-HYDROXY-5-FLUOROPYRIDE-6-ONE-MONOSODIUM SALT AND ITS TAUTOMERS BAYER AG (DE) 2000-01-26 EP disclosed
WO-1998043958-A1 METHOD FOR THE PRODUCTION OF 2,6-DICHLORO-5-FLUORONICOTINONITRILE AND THE CHEMICAL COMPOUND 3-CYANO-2-HYDROXY-5-FLUOROPYRIDE-6-ONE-MONOSODIUM SALT AND ITS TAUTOMERS BAYER AKTIENGESELLSCHAFT (DE) 1998-10-08 WO disclosed