SCHEMBL7896286

SCHEMBL7896286

O=C(c1ccc(C(F)(F)F)cc1)C(F)(F)SC1CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
SRD5A2 P31213 1/20 0.43
HSD11B1 P28845 1/20 0.43
GAA P10253 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
GSK3B P49841 2/20 0.42
PTPN1 P18031 2/20 0.42
MGLL Q99685 1/20 0.42
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM2B Q8NHM5 2/20 0.40
BACE1 P56817 1/20 0.40
NR4A1 P22736 1/20 0.39
NR4A2 P43354 1/20 0.39
NR4A3 Q92570 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7605938 0.85 CES2 (0.41) CES2CES1HSD11B1
SCHEMBL7896288 0.83 CES1 (0.52) CES2CES1HSD11B1GAATSHR
SCHEMBL7609999 0.75 CES2 (0.55) CES2CES1SRD5A2GSK3BPTPN1
SCHEMBL7896290 0.74 CES2 (0.53) CES2CES1SRD5A2HSD11B1GAA
SCHEMBL4023293 0.73 HSD11B1 (0.63) CES2CES1SRD5A2HSD11B1GAA
SCHEMBL6942780 0.72 CES2 (0.52) CES2CES1SRD5A2GSK3BPTPN1
SCHEMBL7886413 0.72 PTPN1 (0.53) CES2CES1SRD5A2HSD11B1GAA
SCHEMBL23172558 0.72 CES2 (0.67) CES2CES1SRD5A2GSK3BPTPN1
SCHEMBL1078685 0.72 CES1 (0.67) CES2CES1SRD5A2GSK3BPTPN1
SCHEMBL1855141 0.70 HSD11B1 (0.60) CES2CES1SRD5A2HSD11B1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6184396-B1 2-CYCLOPROPYLTHIADIFLUOROMETHYL-2-PHENYLOXIRANE INTERMEDIATES FOR 1-(CYCLOPROPYLTHIA)-2-PHENYL-1,1-(CYCLOPROPYLTHIA)-2-PHENYL-1,1-DIFLUORO-3-(1H-1,2,4-TRIAZOL-1-YL)-2-PROPANOL AND DERIVATIVES; FUNGICIDES; CANDIDA AND ASPERGILLUS SSP CO., LTD. (JP) 2001-02-06 US disclosed
US-6172266-B1 FUNGICIDES SSP CO., LTD. (JP) 2001-01-09 US disclosed
US-6040325-A FUNGICIDES FOR THE PREVENTION AND TREATMENT OF MAMMALIAN MYCOTIC INFECTIONS SSP CO., LTD. (JP) 2000-03-21 US disclosed
EP-0933368-A1 Triazole derivative or salt thereof, preparation process thereof and pharmaceutical containing said compound as an effective ingredient (antimycotic) SSP Co., Ltd. (JP) 1999-08-04 EP disclosed