SCHEMBL7899646

SCHEMBL7899646

O=C(CCCc1ccc(Br)cc1)N1CCCC(c2cc3ccccc3[nH]2)C1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
AKR1C3 P42330 1/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GRIN2B Q13224 1/20 0.38
PREP P48147 2/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2789326 0.77 AKR1C3 (0.49) HPGDSMN1; SMN2AKR1C3KDM4E
SCHEMBL7893346 0.73 PROKR1 (0.43) HPGDSMN1; SMN2ALDH1A1MAPK1KDM4E
SCHEMBL8215188 0.70 ADAM17 (0.40) AKR1C3
SCHEMBL14452407 0.70 ADAM17 (0.40) AKR1C3
SCHEMBL13605836 0.70 ADAM17 (0.40) AKR1C3
SCHEMBL7899970 0.70 HPGDS (0.51) HPGDAKR1C3ALDH1A1KDM4E
SCHEMBL2789436 0.70 HPGDS (0.51) HPGDAKR1C3ALDH1A1KDM4E
SCHEMBL2819315 0.69 CYP51A1 (0.37) HPGDSMN1; SMN2ALDH1A1GRIN2B
SCHEMBL27367437 0.68 DRD2 (0.52) AKR1C3KDM4E
SCHEMBL6067790 0.68 HPGD (0.61) HPGDSMN1; SMN2ALDH1A1MAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed