SCHEMBL27367437

SCHEMBL27367437

CN1CCCC(c2cc3ccccc3[nH]2)C1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
KCNH2 Q12809 1/20 0.52
HRH3 Q9Y5N1 3/20 0.46
PARP1 P09874 2/20 0.46
LSS P48449 1/20 0.44
HRH4 Q9H3N8 3/20 0.43
DRD3 P35462 1/20 0.43
CCNT1 O60563 2/20 0.43
CDK9 P50750 2/20 0.43
CHRNA7 P36544 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ATM Q13315 1/20 0.42
AKR1C3 P42330 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
HTR7 P34969 1/20 0.41
ADRA1B P35368 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7203954 0.82 HRH4 (0.53) HTR2AHRH3HRH4CHRNA7HTR7
SCHEMBL20284611 0.81 HRH4 (0.45) DRD2HTR2AHTR2CKCNH2PARP1
SCHEMBL6650886 0.81 DRD2 (0.48) DRD2HTR2AHTR2CKCNH2PARP1
SCHEMBL3640169 0.80 AOC3 (0.44) KDM4EHTR7ADRA1B
SCHEMBL2789326 0.80 AKR1C3 (0.49) HRH3HRH4KDM4EAKR1C3
SCHEMBL2009005 0.79 CCNT1 (0.52) KCNH2HRH3HRH4CCNT1CDK9
SCHEMBL10441226 0.78 AOC3 (0.42) KDM4EHTR7ADRA1B
SCHEMBL13634946 0.77 CHRNB2 (0.50) HTR2AHTR2CKCNH2HRH3PARP1
SCHEMBL73543 0.76 AOC3 (0.47) CHRNA7KDM4E
SCHEMBL7899970 0.76 HPGDS (0.51) PARP1KDM4EAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024059951-A1 INHIBITORS OF THE ANDROGEN RECEPTOR DNA-BINDING DOMAIN THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2024-03-28 WO disclosed