SCHEMBL789995

SCHEMBL789995

N#Cc1cc2cc(Cl)ccc2nc1N

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.62
ALDH1A1 P00352 3/20 0.62
GAA P10253 1/20 0.62
GPR35 Q9HC97 1/20 0.44
CSNK1A1 P48729 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
PSMB8 P28062 3/20 0.42
PSMB5 P28074 1/20 0.42
PIK3CG P48736 2/20 0.42
KHK P50053 1/20 0.41
PKM P14618 1/20 0.40
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807478 0.79 KDM4E (0.62) KDM4EALDH1A1GAAPKMLMNA
SCHEMBL789748 0.79 KDM4E (0.62) KDM4EALDH1A1GAACSNK1A1CLK4
SCHEMBL941858 0.77 ALDH1A1 (1.00) KDM4EALDH1A1GAALMNAMAPT
SCHEMBL29904585 0.77 ALDH1A1 (1.00) KDM4EALDH1A1GAALMNAMAPT
SCHEMBL24091986 0.76 KDM4E (0.57) KDM4EALDH1A1GAAPKMLMNA
SCHEMBL22521377 0.76 KDM4E (0.57) KDM4EALDH1A1GAACSNK1A1PKM
SCHEMBL791113 0.73 PRNP (0.48) PIK3CGLMNACYP1A2MAPTTHRB
SCHEMBL10813766 0.72 ALDH1A1 (0.62) KDM4EALDH1A1GAACSNK1A1CLK4
SCHEMBL9633299 0.71 GPR35 (0.53) KDM4EGPR35PSMB8PSMB5LMNA
SCHEMBL23110066 0.71 ACHE (0.45) KDM4EPSMB8PSMB5PIK3CGLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed