SCHEMBL7901244

SCHEMBL7901244

CCCCOc1cccc2c1cc(C1CCCN(C(=O)C[C@@H](Cc3ccc(Br)cc3)NC(=O)OC(C)(C)C)C1)n2CCCOC

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.34
BCHE P06276 2/20 0.34
CNR2 P34972 3/20 0.34
CACNA1B Q00975 1/20 0.34
HRH2 P25021 4/20 0.34
HRH1 P35367 4/20 0.34
KLK5 Q9Y337 1/20 0.33
PTPN1 P18031 5/20 0.33
F2 P00734 1/20 0.33
PRSS1 P07477 1/20 0.33
REN P00797 1/20 0.32
PTPN22 Q9Y2R2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7896622 0.90 CNR2 (0.35) CNR2CACNA1BHRH2HRH1KLK5
SCHEMBL7891183 0.87 PADI4 (0.40) CNR2CACNA1BHRH2HRH1KLK5
SCHEMBL7896929 0.87 CACNA1B (0.33) CNR2CACNA1BHRH2HRH1KLK5
SCHEMBL7906019 0.86 PDE2A (0.34) CNR2CACNA1BHRH2HRH1KLK5
SCHEMBL7898758 0.84 CNR2 (0.36) CNR2HRH2HRH1KLK5REN
SCHEMBL7891178 0.84 CNR2 (0.36) CNR2HRH2HRH1KLK5REN
SCHEMBL7899697 0.83 PROKR1 (0.39) CNR2CACNA1BHRH2HRH1KLK5
SCHEMBL7901247 0.82 CNR2 (0.33) CNR2HRH2HRH1KLK5PTPN1
SCHEMBL2789237 0.81 CNR2 (0.37) CNR2REN
SCHEMBL2788383 0.81 KLK5 (0.36) CNR2CACNA1BHRH2HRH1KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed