SCHEMBL7906019

SCHEMBL7906019

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc(Br)cc3)NC(=O)OC(C)(C)C)C2)cc2c(OC)nccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.34
PDE3A Q14432 1/20 0.34
HRH2 P25021 4/20 0.33
HRH1 P35367 4/20 0.33
CACNA1B Q00975 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
KLK5 Q9Y337 1/20 0.33
CNR2 P34972 2/20 0.32
FPR2 P25090 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
CCNK O75909 1/20 0.31
CDK12 Q9NYV4 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
PADI4 Q9UM07 1/20 0.31
ACE P12821 1/20 0.31
DYRK1A Q13627 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7896929 0.93 CACNA1B (0.33) PDE2APDE3AHRH2HRH1CACNA1B
SCHEMBL7901623 0.90 ALOX5AP (0.33) PDE2APDE3AHRH2HRH1CCNT1
SCHEMBL7896622 0.87 CNR2 (0.35) HRH2HRH1CACNA1BKLK5CNR2
SCHEMBL7891183 0.87 PADI4 (0.40) HRH2HRH1CACNA1BKLK5CNR2
SCHEMBL7901244 0.86 HTR6 (0.34) HRH2HRH1CACNA1BKLK5CNR2
SCHEMBL7901932 0.81 PTGS2 (0.34) HRH2HRH1CACNA1BKLK5CNR2
SCHEMBL7891178 0.81 CNR2 (0.36) HRH2HRH1KLK5CNR2PADI4
SCHEMBL7898758 0.81 CNR2 (0.36) HRH2HRH1KLK5CNR2PADI4
SCHEMBL7898298 0.81 WNT3A (0.32) PDE2APDE3AHRH2HRH1CCNT1
SCHEMBL7899697 0.81 PROKR1 (0.39) HRH2HRH1CACNA1BKLK5CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed