Bromide

Bromide

SCHEMBL7902023

COC(=O)c1ccc(O)c(C[P+](c2ccccc2)(c2ccccc2)c2ccccc2)c1.[Br-]

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA12 O43570 1/20 0.50
CA7 P43166 1/20 0.50
XDH P47989 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
HPGD P15428 3/20 0.48
ALDH1A1 P00352 2/20 0.48
TP53 P04637 2/20 0.48
ALOX15 P16050 2/20 0.48
ALOX12 P18054 2/20 0.48
HSD17B10 Q99714 2/20 0.48
HIF1A Q16665 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
CKS1B P61024 1/20 0.48
SKP2 Q13309 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7524637 0.97 CA1 (0.50) CA1CA2CA12CA7XDH
Bromide SCHEMBL7898722 0.89 XDH (0.50) CA1CA2CA12CA7XDH
Bromide SCHEMBL11599708 0.86 KDM4E (0.49) HPGDALDH1A1HSD17B10LMNAMAPT
Bromide SCHEMBL7292931 0.83 MAPT (0.47) HPGDALDH1A1HSD17B10HIF1ALMNA
Bromide SCHEMBL8899989 0.83 P4HB (0.46) CA1CA2CA12CA7XDH
Bromide SCHEMBL8901631 0.83 PPARG (0.43) ALDH1A1CYP1A2CYP2C19MAPTMEN1
Bromide SCHEMBL8323844 0.83 DPP4 (0.47) CA1CA2CA12CA7XDH
Bromide SCHEMBL10980300 0.83 KDM4E (0.49) HPGDALDH1A1ALOX15HSD17B10LMNA
SCHEMBL8408482 0.79 HPGD (0.70) CA1CA2CA12CA7XDH
Bromide SCHEMBL2316144 0.79 VCAM1 (0.49) HPGDALDH1A1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194450-B1 KERATINIZATION DISORDERS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2001-02-27 US disclosed
US-5849798-A Polyaromatic heterocyclic compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 1998-12-15 US disclosed