SCHEMBL7903015

SCHEMBL7903015

COC(=O)c1cc2c(nc1C)C(Cl)CCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.44
PFKFB3 Q16875 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK4 Q16654 1/20 0.40
GAA P10253 1/20 0.39
OPRK1 P41145 3/20 0.39
KDM4E B2RXH2 3/20 0.39
KMT2A Q03164 3/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPT P10636 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7911302 0.96 ACHE (0.46) ACHEPFKFB3PDK2PDK4GAA
SCHEMBL7910219 0.87 KDM4E (0.49) ACHEGAAOPRK1KDM4EKMT2A
SCHEMBL7913218 0.85 ACHE (0.42) ACHEPFKFB3PDK2PDK4GAA
SCHEMBL7902939 0.84 KDM4E (0.51) ACHEGAAOPRK1KDM4EKMT2A
SCHEMBL7912964 0.82 ACHE (0.44) ACHEPDK2PDK4GAAOPRK1
SCHEMBL8132938 0.79 SLC9A1 (0.36)
SCHEMBL927361 0.79 ACHE (0.41) ACHEPDK2PDK4GAAOPRK1
SCHEMBL927301 0.78 ACHE (0.41) ACHEPDK2PDK4GAAOPRK1
SCHEMBL7913174 0.76 SLC9A1 (0.38) ACHEKDM4ERAB9AALDH1A1MAPT
SCHEMBL927383 0.75 OPRK1 (0.39) ACHEPDK2PDK4GAAOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6258829-B1 ANTIARRTHMIA AGENTS AND CARDIOVASCULAR DISORDERS TOA EIYO LTD. (JP) 2001-07-10 US disclosed
EP-0972767-A1 CYCLOALKA[b]PYRIDINE-3-CARBONYLGUANIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND DRUGS CONTAINING THE SAME TOA EIYO LTD. (JP) 2000-01-19 EP disclosed