SCHEMBL7904485

SCHEMBL7904485

CCc1cc(C(=O)NC(C)(C)C)ccc1S(=O)(=O)n1nc(OC)n(C2CC2)c1=O

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
DHODH Q02127 1/20 0.34
AVPR1A P37288 1/20 0.34
ANO1 Q5XXA6 2/20 0.33
USP2 O75604 2/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
KDM1A O60341 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
RORC P51449 3/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PDE7A Q13946 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16167675 0.89 ALDH1A1 (0.39) ALDH1A1DHODHAVPR1AANO1LMNA
SCHEMBL16167674 0.81 AVPR1A (0.37) ALDH1A1DHODHAVPR1AUSP2LMNA
SCHEMBL7911467 0.80 ALDH1A1 (0.39) ALDH1A1AVPR1ALMNAHTTPOLB
SCHEMBL7908197 0.79 ALDH1A1 (0.38) ALDH1A1AVPR1ALMNAMAPTKMT2A
SCHEMBL7909327 0.78 AVPR1A (0.39) ALDH1A1OPRM1OPRD1DHODHAVPR1A
SCHEMBL7914828 0.78 AVPR1A (0.39) ALDH1A1AVPR1ALMNAMAPTKMT2A
SCHEMBL7909318 0.78 AVPR1A (0.37) ALDH1A1DHODHAVPR1ALMNAMAPT
SCHEMBL7908194 0.78 KMT2A (0.38) ALDH1A1AVPR1ALMNAMAPTKMT2A
SCHEMBL16167673 0.77 HSD11B1 (0.40) ALDH1A1AVPR1AHTTKMT2A
SCHEMBL2511918 0.69 HSD11B1 (0.46) ALDH1A1LMNAHTTPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063402-A1 SUBSTITUTED BENZYL AND PHENYLSULFONYL TRIAZOLONES, AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-06-10 WO disclosed